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  4. Structure-Based Design of New Pyrazole Inhibitors Targeting Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH)

Structure-Based Design of New Pyrazole Inhibitors Targeting Plasmodium falciparum dihydroorotate dehydrogenase (PfDHODH)

Date

2026

Authors

Agnese Chiara Pippione
Noemi Villella
Federico Fornaseri
Marta Giorgis
Manmohan Sharma
Barbara Rolando
Stefano Sainas
Efrain Salamanca
Alberto Gimenez
Sandrine Cojean

Journal Title

Journal ISSN

Volume Title

Publisher

Elsevier BV

Abstract

Description

Keywords

Chemistry, Dihydroorotate dehydrogenase, Plasmodium falciparum, Pyrazole, Biochemistry, Enzyme, Enzyme inhibitor, In vitro, Stereochemistry, Malaria

Citation

DOI

10.1016/j.ejmech.2026.118753

URI

https://doi.org/10.1016/j.ejmech.2026.118753
https://andeanlibrary.org/handle/123456789/79961

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